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3ENE

Complex of PI3K gamma with an inhibitor

Summary for 3ENE
Entry DOI10.2210/pdb3ene/pdb
DescriptorPhosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, 1-methyl-3-naphthalen-2-yl-1H-pyrazolo[3,4-d]pyrimidin-4-amine (3 entities in total)
Functional Keywordslipid kinase, phosphoinositide, inhibitor, 3-kinase, signaling, pyrazolopyrimidine, pik-208, s2, kinase, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight110071.37
Authors
Apsel, B.,Blair, J.A.,Gonzalez, B.Z.,Nazif, T.M.,Feldman, M.E.,Williams, R.L.,Shokat, K.M.,Knight, Z.A. (deposition date: 2008-09-25, release date: 2008-10-14, Last modification date: 2023-11-01)
Primary citationApsel, B.,Blair, J.A.,Gonzalez, B.,Nazif, T.M.,Feldman, M.E.,Aizenstein, B.,Hoffman, R.,Williams, R.L.,Shokat, K.M.,Knight, Z.A.
Targeted polypharmacology: discovery of dual inhibitors of tyrosine and phosphoinositide kinases
Nat.Chem.Biol., 4:691-699, 2008
Cited by
PubMed: 18849971
DOI: 10.1038/nchembio.117
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

217705

數據於2024-03-27公開中

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