3DSE
A potent peptidomimetic inhibitor of botulinum neurotoxin serotype A has a very different conformation than SNAP-25 substrate
Summary for 3DSE
Entry DOI | 10.2210/pdb3dse/pdb |
Related | 1XTF 2ISG 3DS9 3DSE |
Descriptor | Botulinum neurotoxin type A, ZINC ION, NICKEL (II) ION, ... (4 entities in total) |
Functional Keywords | snare, botulism, inhibition, metalloprotease, neurotransmission, neuromuscular junction, hydrolase, membrane, metal-binding, neurotoxin, pharmaceutical, protease, secreted, toxin, transmembrane, zinc |
Biological source | Clostridium botulinum |
Cellular location | Botulinum neurotoxin A light chain: Secreted. Botulinum neurotoxin A heavy chain: Secreted: A5HZZ9 |
Total number of polymer chains | 1 |
Total formula weight | 47902.09 |
Authors | Zuniga, J.E.,Fenn, T. (deposition date: 2008-07-11, release date: 2008-09-30, Last modification date: 2024-02-21) |
Primary citation | Zuniga, J.E.,Schmidt, J.J.,Fenn, T.,Burnett, J.C.,Arac, D.,Gussio, R.,Stafford, R.G.,Badie, S.S.,Bavari, S.,Brunger, A.T. A Potent Peptidomimetic Inhibitor of Botulinum Neurotoxin Serotype A Has a Very Different Conformation than SNAP-25 Substrate Structure, 16:1588-1597, 2008 Cited by PubMed: 18940613DOI: 10.1016/j.str.2008.07.011 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
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