3DLS
Crystal structure of human PAS kinase bound to ADP
3DLS の概要
エントリーDOI | 10.2210/pdb3dls/pdb |
分子名称 | PAS domain-containing serine/threonine-protein kinase, MAGNESIUM ION, ADENOSINE-5'-DIPHOSPHATE, ... (4 entities in total) |
機能のキーワード | pas kinase, pask, protein kinase, drug discovery, atp-binding, kinase, nucleotide-binding, phosphoprotein, serine/threonine-protein kinase, transferase, structural genomics, psi-2, protein structure initiative, new york sgx research center for structural genomics, nysgxrc |
由来する生物種 | Homo sapiens (Human) |
タンパク質・核酸の鎖数 | 6 |
化学式量合計 | 230276.62 |
構造登録者 | Antonysamy, S.,Bonanno, J.B.,Romero, R.,Russell, M.,Iizuka, M.,Gheyi, T.,Wasserman, S.R.,Rutter, J.,Sauder, J.M.,Burley, S.K.,New York SGX Research Center for Structural Genomics (NYSGXRC) (登録日: 2008-06-29, 公開日: 2008-08-26, 最終更新日: 2024-02-21) |
主引用文献 | Kikani, C.K.,Antonysamy, S.A.,Bonanno, J.B.,Romero, R.,Zhang, F.F.,Russell, M.,Gheyi, T.,Iizuka, M.,Emtage, S.,Sauder, J.M.,Turk, B.E.,Burley, S.K.,Rutter, J. Structural bases of PAS domain-regulated kinase (PASK) activation in the absence of activation loop phosphorylation. J.Biol.Chem., 285:41034-41043, 2010 Cited by PubMed: 20943661DOI: 10.1074/jbc.M110.157594 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.3 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード