3CDM
Structural adaptation and conservation in quadruplex-drug recognition
Summary for 3CDM
Entry DOI | 10.2210/pdb3cdm/pdb |
Related | 3CCO |
Descriptor | DNA (5'-D(*DT*DAP*DGP*DGP*DGP*DTP*DTP*DAP*DGP*DGP*DGP*DTP*DTP*DAP*DGP*DGP*DGP*DTP*DTP*DAP*DGP*DGP*DG)-3'), 2,7-bis[3-(dimethylamino)propyl]-4,9-bis[(3-hydroxypropyl)amino]benzo[lmn][3,8]phenanthroline-1,3,6,8(2H,7H)-tetrone, POTASSIUM ION, ... (4 entities in total) |
Functional Keywords | quadruplex, dna, propeller, intramolecular, human telomere parallel stranded, ligand, complex |
Total number of polymer chains | 2 |
Total formula weight | 18227.92 |
Authors | Parkinson, G.N.,Neidle, S. (deposition date: 2008-02-27, release date: 2008-09-23, Last modification date: 2023-11-01) |
Primary citation | Parkinson, G.N.,Cuenca, F.,Neidle, S. Topology conservation and loop flexibility in quadruplex-drug recognition: crystal structures of inter- and intramolecular telomeric DNA quadruplex-drug complexes J.Mol.Biol., 381:1145-1156, 2008 Cited by PubMed: 18619463DOI: 10.1016/j.jmb.2008.06.022 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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