3B1M
Crystal structure of the PPARgamma-LBD complexed with a cercosporamide derivative modulator Cerco-A
Summary for 3B1M
Entry DOI | 10.2210/pdb3b1m/pdb |
Related | 3LMP |
Descriptor | Peroxisome proliferator-activated receptor gamma, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, (9aS)-8-acetyl-N-[(2-ethylnaphthalen-1-yl)methyl]-1,7-dihydroxy-3-methoxy-9a-methyl-9-oxo-9,9a-dihydrodibenzo[b,d]furan-4-carboxamide, ... (4 entities in total) |
Functional Keywords | transcription |
Biological source | Homo sapiens (human) More |
Cellular location | Nucleus: P37231 Q9UBK2 |
Total number of polymer chains | 2 |
Total formula weight | 34993.50 |
Authors | Matsui, Y.,Hiroyuki, H. (deposition date: 2011-07-05, release date: 2011-08-24, Last modification date: 2023-11-01) |
Primary citation | Wakabayashi, K.,Hayashi, S.,Matsui, Y.,Matsumoto, T.,Furukawa, A.,Kuroha, M.,Tanaka, N.,Inaba, T.,Kanda, S.,Tanaka, J.,Okuyama, R.,Wakimoto, S.,Ogata, T.,Araki, K.,Ohsumi, J. Pharmacology and in Vitro Profiling of a Novel Peroxisome Proliferator-Activated Receptor gamma Ligand, Cerco-A Biol.Pharm.Bull., 34:1094-1104, 2011 Cited by PubMed: 21720019DOI: 10.1248/bpb.34.1094 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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