Summary for 3HVC
Entry DOI | 10.2210/pdb3hvc/pdb |
Descriptor | Mitogen-activated protein kinase 14, 4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDINE (3 entities in total) |
Functional Keywords | transferase, map kinase, serine/threonine-protein kinase, p38, isoform-2, alternative splicing, atp-binding, cytoplasm, kinase, nucleotide-binding, nucleus, phosphoprotein, polymorphism |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm (By similarity): Q16539 |
Total number of polymer chains | 1 |
Total formula weight | 41975.86 |
Authors | Perry, J.J.,Tainer, J.A. (deposition date: 2009-06-15, release date: 2009-06-30, Last modification date: 2023-09-06) |
Primary citation | Perry, J.J.,Harris, R.M.,Moiani, D.,Olson, A.J.,Tainer, J.A. p38alpha MAP kinase C-terminal domain binding pocket characterized by crystallographic and computational analyses. J.Mol.Biol., 391:1-11, 2009 Cited by PubMed: 19501598DOI: 10.1016/j.jmb.2009.06.005 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
Download full validation report