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2ZJW

Crystal structure of human CK2 alpha complexed with Ellagic acid

Summary for 2ZJW
Entry DOI10.2210/pdb2zjw/pdb
DescriptorCasein kinase II subunit alpha, 2,3,7,8-tetrahydroxychromeno[5,4,3-cde]chromene-5,10-dione (3 entities in total)
Functional Keywordsprotein-inhibitor complex, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase, wnt signaling pathway
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight40780.38
Authors
Sekiguchi, Y.,Kinoshita, T.,Nakaniwa, T.,Tada, T. (deposition date: 2008-03-11, release date: 2009-03-17, Last modification date: 2023-11-01)
Primary citationSekiguchi, Y.,Nakaniwa, T.,Kinoshita, T.,Nakanishi, I.,Kitaura, K.,Hirasawa, A.,Tsujimoto, G.,Tada, T.
Structural insight into human CK2alpha in complex with the potent inhibitor ellagic acid
Bioorg.Med.Chem.Lett., 19:2920-2923, 2009
Cited by
PubMed: 19414254
DOI: 10.1016/j.bmcl.2009.04.076
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

217705

건을2024-03-27부터공개중

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