2VD5
Structure of Human Myotonic Dystrophy Protein Kinase in Complex with the Bisindoylmaleide inhibitor BIM VIII
Summary for 2VD5
Entry DOI | 10.2210/pdb2vd5/pdb |
Descriptor | DMPK PROTEIN, 3-[1-(3-AMINOPROPYL)-1H-INDOL-3-YL]-4-(1-METHYL-1H-INDOL-3-YL)-1H-PYRROLE-2,5-DIONE (3 entities in total) |
Functional Keywords | serine/threonine-protein kinase, kinase, transferase, atp-binding, nucleotide-binding, cardiac contractility, muscle differentiation |
Biological source | HOMO SAPIENS (HUMAN) |
Total number of polymer chains | 2 |
Total formula weight | 93007.64 |
Authors | Pike, A.C.W.,Amos, A.,Elkins, J.,Bullock, A.,Guo, K.,Fedorov, O.,Bunkoczi, G.,Filippakopoulos, P.,Pilka, E.S.,Ugochukwu, E.,Umeano, C.,Niesen, F.,Sundstrom, M.,Weigelt, J.,Edwards, A.,Arrowsmith, C.H.,von Delft, F.,Knapp, S. (deposition date: 2007-09-30, release date: 2007-11-06, Last modification date: 2023-12-13) |
Primary citation | Elkins, J.,Amos, A.,Niesen, F.,Pike, A.C.W.,Fedorov, O.,Knapp, S. Structure of Dystrophia Myotonica Protein Kinase. Protein Sci., 18:782-, 2009 Cited by PubMed: 19309729DOI: 10.1002/PRO.82 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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