2RD4
Design of specific inhibitors of Phospholipase A2: Crystal structure of the complex of phospholipase A2 with pentapeptide Leu-Val-Phe-Phe-Ala at 2.9 A resolution
2RD4 の概要
| エントリーDOI | 10.2210/pdb2rd4/pdb |
| 関連するPDBエントリー | 1S6B |
| 分子名称 | Phospholipase A2 isoform 1, Phospholipase A2 isoform 2, pentapeptide inhibitor, ... (5 entities in total) |
| 機能のキーワード | phospholipase a2, peptide inhibitor, complex, calcium, hydrolase, lipid degradation, metal-binding, secreted |
| 由来する生物種 | Naja sagittifera 詳細 |
| 細胞内の位置 | Secreted: P60043 P60044 |
| タンパク質・核酸の鎖数 | 3 |
| 化学式量合計 | 27185.25 |
| 構造登録者 | Mirza, Z.,Kaur, A.,Singh, N.,Sinha, M.,Sharma, S.,Srinivasan, A.,Kaur, P.,Singh, T.P. (登録日: 2007-09-21, 公開日: 2007-10-09, 最終更新日: 2024-11-06) |
| 主引用文献 | Mirza, Z.,Kaur, A.,Singh, N.,Sinha, M.,Sharma, S.,Srinivasan, A.,Kaur, P.,Singh, T.P. Design of specific inhibitors of Phospholipase A2: Crystal structure of the complex of phospholipase A2 with pentapeptide Leu-Val-Phe-Phe-Ala at 2.9 A resolution To be Published, |
| 実験手法 | X-RAY DIFFRACTION (2.97 Å) |
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