2QPY

AR LBD with small molecule

Summary for 2QPY

Entry DOI	10.2210/pdb2qpy/pdb
Descriptor	Androgen receptor, Coactivator peptide, 5-ALPHA-DIHYDROTESTOSTERONE, ... (5 entities in total)
Functional Keywords	androgen receptor dht coactivator, dna-binding, lipid-binding, metal-binding, nucleus, steroid-binding, transcription, transcription regulation, ubl conjugation, zinc, zinc-finger, dna binding protein
Biological source	Mus musculus (house mouse) More
Cellular location	Nucleus : P19091
Total number of polymer chains	2
Total formula weight	31455.17
Authors	Estebanez-Perpina, E.,Fletterick, R. (deposition date: 2007-07-25, release date: 2007-09-25, Last modification date: 2024-02-21)
Primary citation	Estebanez-Perpina, E.,Arnold, L.A.,Arnold, A.A.,Nguyen, P.,Rodrigues, E.D.,Mar, E.,Bateman, R.,Pallai, P.,Shokat, K.M.,Baxter, J.D.,Guy, R.K.,Webb, P.,Fletterick, R.J. A surface on the androgen receptor that allosterically regulates coactivator binding. Proc.Natl.Acad.Sci.Usa, 104:16074-16079, 2007 Cited by PubMed: 17911242 DOI: 10.1073/pnas.0708036104 PDB entries with the same primary citation
Experimental method	X-RAY DIFFRACTION (2.5 Å)

Structure validation