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2QLN

Glycogen Phosphorylase b in complex with N-4-phenylbenzoyl-N'-beta-D-glucopyranosyl urea

2QLN の概要
エントリーDOI10.2210/pdb2qln/pdb
関連するPDBエントリー2QLM 2QN3 2QN7 2QN8 2QN9 2QNB
分子名称Glycogen phosphorylase, muscle form, N-[(biphenyl-4-ylcarbonyl)carbamoyl]-beta-D-glucopyranosylamine (3 entities in total)
機能のキーワードglycogenolysis, type 2 diabetes, acetylation, allosteric enzyme, carbohydrate metabolism, glycogen metabolism, glycosyltransferase, nucleotide-binding, phosphoprotein, pyridoxal phosphate, transferase
由来する生物種Oryctolagus cuniculus (Rabbit)
タンパク質・核酸の鎖数1
化学式量合計97921.72
構造登録者
Oikonomakos, N.G.,Chrysina, E.D.,Tiraidis, C.,Alexacou, K.-M.,Leonidas, D.D.,Sographos, S.E. (登録日: 2007-07-13, 公開日: 2008-07-15, 最終更新日: 2023-11-15)
主引用文献Nagy, V.,Felf ldi, N.,Praly, J.-P.,Dosca, T.,Gergerly, P.,Chrysina, E.D.,Tiraidis, C.,Kosmopoulou, M.N.,Alexacou, K.-M.,Konstantakaki, M.
N-(4-substituted-benzoyl)-N'-(beta-D-glucopyranosyl)ureas, inhibitors of glycogen phosphorylase: synthesis, kinetic and crystallographic evaluation
To be Published,
実験手法
X-RAY DIFFRACTION (2.15 Å)
構造検証レポート
Validation report summary of 2qln
検証レポート(詳細版)ダウンロードをダウンロード

217705

件を2024-03-27に公開中

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