2PH9
Galanthamine bound to an ACh-binding Protein
Summary for 2PH9
Entry DOI | 10.2210/pdb2ph9/pdb |
Related | 2PGZ |
Descriptor | Soluble acetylcholine receptor, (-)-GALANTHAMINE, TETRAETHYLENE GLYCOL, ... (4 entities in total) |
Functional Keywords | non-competitive inhibitors, nicotinic acetylcholine receptor, acetylcholine-binding protein, benzodiazepine, galanthamine, choline-binding protein |
Biological source | Aplysia californica (California sea hare) |
Total number of polymer chains | 5 |
Total formula weight | 132404.17 |
Authors | Hansen, S.B.,Taylor, P. (deposition date: 2007-04-10, release date: 2007-07-03, Last modification date: 2023-08-30) |
Primary citation | Hansen, S.B.,Taylor, P. Galanthamine and non-competitive inhibitor binding to ACh-binding protein: evidence for a binding site on non-alpha-subunit interfaces of heteromeric neuronal nicotinic receptors. J.Mol.Biol., 369:895-901, 2007 Cited by PubMed: 17481657DOI: 10.1016/j.jmb.2007.03.067 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.88 Å) |
Structure validation
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