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2N27

Competitive inhibition of TRPV1 calmodulin interaction by vanilloids

Summary for 2N27
Entry DOI10.2210/pdb2n27/pdb
NMR InformationBMRB: 25588
DescriptorCalmodulin, CALCIUM ION, (6E)-N-(4-hydroxy-3-methoxybenzyl)-8-methylnon-6-enamide (3 entities in total)
Functional Keywordscalmodulin, capsaicin, metal binding protein
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm, cytoskeleton, spindle : P62158
Total number of polymer chains1
Total formula weight17187.07
Authors
Hetenyi, A.,Nemeth, L.,Weber, E.,Szakonyi, G.,Winter, Z.,Josvay, K.,Bartus, E.,Olah, Z.,Martinek, T.A. (deposition date: 2015-04-29, release date: 2016-07-06, Last modification date: 2023-06-14)
Primary citationHetenyi, A.,Nemeth, L.,Weber, E.,Szakonyi, G.,Winter, Z.,Josvay, K.,Bartus, E.,Olah, Z.,Martinek, T.A.
Competitive inhibition of TRPV1-calmodulin interaction by vanilloids.
Febs Lett., 590:2768-2775, 2016
Cited by
PubMed: 27339229
DOI: 10.1002/1873-3468.12267
PDB entries with the same primary citation
Experimental method
SOLUTION NMR
Structure validation

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