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2JBK

membrane-bound glutamate carboxypeptidase II (GCPII) in complex with quisqualic acid (quisqualate, alpha-amino-3,5-dioxo-1,2,4- oxadiazolidine-2-propanoic acid)

2JBK の概要
エントリーDOI10.2210/pdb2jbk/pdb
関連するPDBエントリー1Z8L 2C6C 2C6G 2C6P 2CIJ 2JBJ
分子名称GLUTAMATE CARBOXYPEPTIDASE 2, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (9 entities in total)
機能のキーワードmultifunctional enzyme, neurodegenerative disease, glycoprotein, metal-binding, signal-anchor, hydrolase, naaladase, dipeptidase, polymorphism, zinc, psma, antigen, membrane, protease, peptidase, transmembrane, metal- binding, metalloprotease, prostate cancer, carboxypeptidase
由来する生物種HOMO SAPIENS (HUMAN)
タンパク質・核酸の鎖数1
化学式量合計82695.73
構造登録者
Mesters, J.R.,Henning, K.,Hilgenfeld, R. (登録日: 2006-12-07, 公開日: 2006-12-18, 最終更新日: 2023-12-13)
主引用文献Mesters, J.R.,Henning, K.,Hilgenfeld, R.
Human Glutamate Carboxypeptidase II Inhibition: Structures of Gcpii in Complex with Two Potent Inhibitors, Quisqualate and 2-Pmpa.
Acta Crystallogr.,Sect.D, 63:508-, 2007
Cited by
PubMed: 17372356
DOI: 10.1107/S090744490700902X
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2.99 Å)
構造検証レポート
Validation report summary of 2jbk
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-09-18に公開中

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