2HNY
Crystal Structure of E138K Mutant HIV-1 Reverse Transcriptase in Complex with Nevirapine
Summary for 2HNY
Entry DOI | 10.2210/pdb2hny/pdb |
Descriptor | Reverse transcriptase/ribonuclease H, PHOSPHATE ION, MAGNESIUM ION, ... (6 entities in total) |
Functional Keywords | hiv-1 reverse transcriptase, aids, non-nucleoside inhibitor, nevirapine, drug resistance mutations, drug design, transferase |
Biological source | Human immunodeficiency virus 1 More |
Cellular location | Matrix protein p17: Virion (Potential). Capsid protein p24: Virion (Potential). Nucleocapsid protein p7: Virion (Potential). Reverse transcriptase/ribonuclease H: Virion (Potential). Integrase: Virion (Potential): P04585 P04585 |
Total number of polymer chains | 2 |
Total formula weight | 111943.28 |
Authors | Ren, J.,Nichols, C.E.,Stamp, A.,Chamberlain, P.P.,Stammers, D.K. (deposition date: 2006-07-13, release date: 2006-09-05, Last modification date: 2021-10-20) |
Primary citation | Ren, J.,Nichols, C.E.,Stamp, A.,Chamberlain, P.P.,Ferris, R.,Weaver, K.L.,Short, S.A.,Stammers, D.K. Structural insights into mechanisms of non-nucleoside drug resistance for HIV-1 reverse transcriptases mutated at codons 101 or 138. Febs J., 273:3850-3860, 2006 Cited by PubMed: 16911530DOI: 10.1111/j.1742-4658.2006.05392.x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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