2CDZ
CRYSTAL STRUCTURE OF THE HUMAN P21-ACTIVATED KINASE 4 IN COMPLEX WITH CGP74514A
Summary for 2CDZ
Entry DOI | 10.2210/pdb2cdz/pdb |
Related | 2BVA |
Descriptor | SERINE/THREONINE-PROTEIN KINASE PAK 4, N2-[(1R,2S)-2-AMINOCYCLOHEXYL]-N6-(3-CHLOROPHENYL)-9-ETHYL-9H-PURINE-2,6-DIAMINE, SULFATE ION, ... (5 entities in total) |
Functional Keywords | transferase, protein kinase, ste20, pak4, atp-binding |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cytoplasm : O96013 |
Total number of polymer chains | 1 |
Total formula weight | 34849.16 |
Authors | Debreczeni, J.E.,Ugochukwu, E.,Eswaran, J.,Filippakopoulos, P.,Das, S.,Fedorov, O.,Sundstrom, M.,Arrowsmith, C.,Weigelt, J.,Edwards, A.,von Delft, F.,Knapp, S. (deposition date: 2006-01-31, release date: 2006-02-08, Last modification date: 2023-12-13) |
Primary citation | Eswaran, J.,Lee, W.H.,Debreczeni, J.E.,Filippakopoulos, P.,Turnbull, A.,Fedorov, O.,Deacon, S.W.,Peterson, J.R.,Knapp, S. Crystal Structures of the P21-Activated Kinases Pak4, Pak5, and Pak6 Reveal Catalytic Domain Plasticity of Active Group II Paks. Structure, 15:201-, 2007 Cited by PubMed: 17292838DOI: 10.1016/J.STR.2007.01.001 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
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