2ZK4
Human peroxisome proliferator-activated receptor gamma ligand binding domain complexed with 15-oxo-eicosatetraenoic acid
Summary for 2ZK4
Entry DOI | 10.2210/pdb2zk4/pdb |
Related | 2ZK0 2ZK1 2ZK2 2ZK3 2ZK5 2ZK6 |
Descriptor | Peroxisome proliferator-activated receptor gamma, (5E,8E,11Z,13E)-15-oxoicosa-5,8,11,13-tetraenoic acid (3 entities in total) |
Functional Keywords | anti parallel helix sandwich, activator, alternative splicing, diabetes mellitus, disease mutation, dna-binding, metal-binding, nucleus, obesity, phosphoprotein, polymorphism, receptor, transcription, transcription regulation, zinc, zinc-finger |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: P37231 |
Total number of polymer chains | 2 |
Total formula weight | 65698.20 |
Authors | Waku, T.,Shiraki, T.,Oyama, T.,Fujimoto, Y.,Morikawa, K. (deposition date: 2008-03-12, release date: 2009-02-24, Last modification date: 2023-11-01) |
Primary citation | Waku, T.,Shiraki, T.,Oyama, T.,Fujimoto, Y.,Maebara, K.,Kamiya, N.,Jingami, H.,Morikawa, K. Structural insight into PPARgamma activation through covalent modification with endogenous fatty acids J.Mol.Biol., 385:188-199, 2009 Cited by PubMed: 18977231DOI: 10.1016/j.jmb.2008.10.039 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.57 Å) |
Structure validation
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