2WIL
AGED FORM OF HUMAN BUTYRYLCHOLINESTERASE INHIBITED BY TABUN ANALOGUE TA5
Summary for 2WIL
Entry DOI | 10.2210/pdb2wil/pdb |
Related | 1EHO 1EHQ 1KCJ 1P0I 1P0M 1P0P 1P0Q 1XLU 1XLV 1XLW 2J4C 2WID 2WIF 2WIG 2WIJ 2WIK |
Descriptor | CHOLINESTERASE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ethylphosphoramidic acid, ... (7 entities in total) |
Functional Keywords | aging, hydrolase, inhibition, polymorphism, glycoprotein, serine esterase, disease mutation |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 123554.10 |
Authors | Carletti, E.,Aurbek, N.,Gillon, E.,Loiodice, M.,Nicolet, Y.,Fontecilla, J.,Masson, P.,Thiermann, H.,Nachon, F.,Worek, F. (deposition date: 2009-05-12, release date: 2009-05-26, Last modification date: 2023-12-13) |
Primary citation | Carletti, E.,Aurbek, N.,Gillon, E.,Loiodice, M.,Nicolet, Y.,Fontecilla, J.,Masson, P.,Thiermann, H.,Nachon, F.,Worek, F. Structure-Activity Analysis of Aging and Reactivation of Human Butyrylcholinesterase Inhibited by Analogues of Tabun Biochem.J., 421:97-, 2009 Cited by PubMed: 19368529DOI: 10.1042/BJ20090091 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.1 Å) |
Structure validation
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