2IEO
Crystal structure analysis of HIV-1 protease mutant I84V with a potent non-peptide inhibitor (UIC-94017)
Replaces: 1S6SSummary for 2IEO
Entry DOI | 10.2210/pdb2ieo/pdb |
Related | 2IDW 2IEN |
Descriptor | Protease, CHLORIDE ION, SODIUM ION, ... (5 entities in total) |
Functional Keywords | hiv-1 protease, mutant, i84v, dimer, inhibitor, uic-94017, tmc114, darunavir, hydrolase |
Biological source | Human immunodeficiency virus 1 |
Total number of polymer chains | 2 |
Total formula weight | 22130.31 |
Authors | Tie, Y.,Boross, P.I.,Wang, Y.F.,Gaddis, L.,Manna, D.,Hussain, A.K.,Leshchenko, S.,Ghosh, A.K.,Louis, J.M.,Harrison, R.W.,Weber, I.T. (deposition date: 2006-09-19, release date: 2006-10-03, Last modification date: 2023-08-30) |
Primary citation | Tie, Y.,Boross, P.I.,Wang, Y.F.,Gaddis, L.,Hussain, A.K.,Leshchenko, S.,Ghosh, A.K.,Louis, J.M.,Harrison, R.W.,Weber, I.T. High Resolution Crystal Structures of HIV-1 Protease with a Potent Non-Peptide Inhibitor (Uic-94017) Active Against Multi-Drug-Resistant Clinical Strains. J.Mol.Biol., 338:341-352, 2004 Cited by PubMed: 15066436DOI: 10.1016/j.jmb.2004.02.052 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.53 Å) |
Structure validation
Download full validation report