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2HNZ

Crystal Structure of E138K Mutant HIV-1 Reverse Transcriptase in Complex with PETT-2

Summary for 2HNZ
Entry DOI10.2210/pdb2hnz/pdb
DescriptorReverse transcriptase/ribonuclease H, PHOSPHATE ION, 1-[2-(4-ETHOXY-3-FLUOROPYRIDIN-2-YL)ETHYL]-3-(5-METHYLPYRIDIN-2-YL)THIOUREA, ... (4 entities in total)
Functional Keywordshiv-1 reverse transcriptase, aids, non-nucleoside inhibitor, pett-2, drug resistance mutations, drug design, transferase
Biological sourceHuman immunodeficiency virus 1
More
Cellular locationMatrix protein p17: Virion (Potential). Capsid protein p24: Virion (Potential). Nucleocapsid protein p7: Virion (Potential). Reverse transcriptase/ribonuclease H: Virion (Potential). Integrase: Virion (Potential): P04585
Total number of polymer chains2
Total formula weight111892.12
Authors
Ren, J.,Nichols, C.E.,Stamp, A.,Chamberlain, P.P.,Stammers, D.K. (deposition date: 2006-07-13, release date: 2006-09-05, Last modification date: 2021-10-20)
Primary citationRen, J.,Nichols, C.E.,Stamp, A.,Chamberlain, P.P.,Ferris, R.,Weaver, K.L.,Short, S.A.,Stammers, D.K.
Structural insights into mechanisms of non-nucleoside drug resistance for HIV-1 reverse transcriptases mutated at codons 101 or 138.
Febs J., 273:3850-3860, 2006
Cited by
PubMed: 16911530
DOI: 10.1111/j.1742-4658.2006.05392.x
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3 Å)
Structure validation

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