1W22
Crystal structure of inhibited human HDAC8
Summary for 1W22
Entry DOI | 10.2210/pdb1w22/pdb |
Related | 1T64 1T67 1T69 1VKG |
Descriptor | HISTONE DEACETYLASE 8, ZINC ION, POTASSIUM ION, ... (5 entities in total) |
Functional Keywords | hydroxamic acid, chromatin, deacetylation, hdac, hydrolase, nuclear protein, repressor |
Biological source | HOMO SAPIENS |
Cellular location | Nucleus: Q9BY41 |
Total number of polymer chains | 2 |
Total formula weight | 84671.06 |
Authors | Vannini, A.,Volpari, C.,Caroli Casavola, E.,Di Marco, S. (deposition date: 2004-06-25, release date: 2004-09-24, Last modification date: 2023-12-13) |
Primary citation | Vannini, A.,Volpari, C.,Filocamo, G.,Caroli Casavola, E.,Brunetti, M.,Renzoni, D.,Chakravarty, P.,Paolini, C.,De Francesco, R.,Gallinari, P.,Steinckuhler, C.,Di Marco, S. Crystal Structure of a Eukaryotic Zn-Dependent Histone Deacetylase,Human Hdac8,Complexed with a Hydroxamic Acid Inhibitor Proc.Natl.Acad.Sci.USA, 101:15064-, 2004 Cited by PubMed: 15477595DOI: 10.1073/PNAS.0404603101 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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