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1VYQ

Novel inhibitors of Plasmodium Falciparum dUTPase provide a platform for anti-malarial drug design

Summary for 1VYQ
Entry DOI10.2210/pdb1vyq/pdb
DescriptorDEOXYURIDINE 5'-TRIPHOSPHATE NUCLEOTIDOHYDROLASE, 2,3-DEOXY-3-FLUORO-5-O-TRITYLURIDINE (3 entities in total)
Functional Keywordsdrug design, plasmodium falciparum, dutpase, deoxyuridine nucleotidohydrolase, malaria, hydrolase
Biological sourcePLASMODIUM FALCIPARUM
Total number of polymer chains3
Total formula weight60227.05
Authors
Primary citationWhittingham, J.L.,Leal, I.,Nguyen, C.,Kasinathan, G.,Bell, E.,Jones, A.F.,Berry, C.,Benito, A.,Turkenburg, J.P.,Dodson, E.J.,Ruiz Perez, L.M.,Wilkinson, A.J.,Johansson, N.G.,Brun, R.,Gilbert, I.H.,Gonzalez Pacanowska, D.,Wilson, K.S.
Dutpase as a Platform for Antimalarial Drug Design: Structural Basis for the Selectivity of a Class of Nucleoside Inhibitors.
Structure, 13:329-, 2005
Cited by
PubMed: 15698576
DOI: 10.1016/J.STR.2004.11.015
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

217705

數據於2024-03-27公開中

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