1U33
In situ extension as an approach for identifying novel alpha-amylase inhibitors
1U33 の概要
エントリーDOI | 10.2210/pdb1u33/pdb |
関連するPDBエントリー | 1U2Y 1U30 |
分子名称 | Alpha-amylase, pancreatic, 2-acetamido-2-deoxy-beta-D-glucopyranose, 4'-O-METHYL-MALTOSYL-ALPHA (1,4)-(Z, 3S,4S,5R,6R)-3,4,5-TRIHYDROXY-6-HYDROXYMETHYL-PIPERIDIN-2-ONE, ... (6 entities in total) |
機能のキーワード | glycosidase, human pancreatic alpha-amylase, acarbose, inhibitor, glucosidase, enzyme mechanism, hydrolase |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 56758.52 |
構造登録者 | Numao, S.,Li, C.,Damager, I.,Wrodnigg, T.M.,Begum, A.,Overall, C.M.,Brayer, G.D.,Withers, S.G. (登録日: 2004-07-20, 公開日: 2004-09-07, 最終更新日: 2020-11-11) |
主引用文献 | Numao, S.,Damager, I.,Li, C.,Wrodnigg, T.M.,Begum, A.,Overall, C.M.,Brayer, G.D.,Withers, S.G. In Situ Extension as an Approach for Identifying Novel alpha-Amylase Inhibitors. J.Biol.Chem., 279:48282-48291, 2004 Cited by PubMed: 15304511DOI: 10.1074/jbc.M406804200 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.95 Å) |
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