1TOM
ALPHA-THROMBIN COMPLEXED WITH HIRUGEN
1TOM の概要
エントリーDOI | 10.2210/pdb1tom/pdb |
分子名称 | ALPHA-THROMBIN, HIRUGEN, METHYL-PHE-PRO-AMINO-CYCLOHEXYLGLYCINE, ... (5 entities in total) |
機能のキーワード | hydrolase, serine protease, kringle, disease mutation, complex (hydrolase-inhibitor), hydrolase-hydrolase inhibitor complex, blood coagulation-hydrolase inhibitor complex, blood coagulation/hydrolase inhibitor |
由来する生物種 | Hirudo medicinalis (medicinal leech) 詳細 |
細胞内の位置 | Secreted, extracellular space: P00734 P00734 Secreted: P28507 |
タンパク質・核酸の鎖数 | 3 |
化学式量合計 | 35869.90 |
構造登録者 | |
主引用文献 | Lyle, T.A.,Chen, Z.G.,Appleby, S.D.,Freidinger, R.M.,Gardell, S.J.,Lewis, S.D.,Li, Y.,Lyle, E.A.,Lynch, J.J.,Mulichak, A.M.,Ng, A.S.,NaylorOlsen, A.M.,Sanders, W.M. Synthesis, evaluation, and crystallographic analysis of L-371,912: A potent and selective active-site thrombin inhibitor. Bioorg.Med.Chem.Lett., 7:67-72, 1997 Cited by |
実験手法 | X-RAY DIFFRACTION (1.8 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード