1SIV
THREE-DIMENSIONAL STRUCTURE OF A SIV PROTEASE(SLASH)INHIBITOR COMPLEX. IMPLICATIONS FOR THE DESIGN OF HIV-1 AND HIV-2 PROTEASE INHIBITORS
1SIV の概要
エントリーDOI | 10.2210/pdb1siv/pdb |
関連するBIRD辞書のPRD_ID | PRD_000320 |
分子名称 | SIV PROTEASE, methyl N-{(4S,5S)-5-[(L-alanyl-L-alanyl)amino]-4-hydroxy-6-phenylhexanoyl}-L-valyl-L-valinate (3 entities in total) |
機能のキーワード | hydrolase-hydrolase inhibitor complex, acid proteinase, hydrolase/hydrolase inhibitor |
由来する生物種 | Simian immunodeficiency virus |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 22028.61 |
構造登録者 | |
主引用文献 | Zhao, B.,Winborne, E.,Minnich, M.D.,Culp, J.S.,Debouck, C.,Abdel-Meguid, S.S. Three-dimensional structure of a simian immunodeficiency virus protease/inhibitor complex. Implications for the design of human immunodeficiency virus type 1 and 2 protease inhibitors. Biochemistry, 32:13054-13060, 1993 Cited by PubMed: 8241159DOI: 10.1021/bi00211a015 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.5 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード