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1P8J

CRYSTAL STRUCTURE OF THE PROPROTEIN CONVERTASE FURIN

Summary for 1P8J
Entry DOI10.2210/pdb1p8j/pdb
Related PRD IDPRD_000278
DescriptorFurin precursor, DECANOYL-ARG-VAL-LYS-ARG-CHLOROMETHYLKETONE INHIBITOR, beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-[beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)]alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... (8 entities in total)
Functional Keywordsprohormone convertase, spc1, pace, p-domain, chloromethylketone, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceMus musculus (house mouse)
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Total number of polymer chains16
Total formula weight426622.72
Authors
Henrich, S.,Cameron, A.,Bourenkov, G.P.,Kiefersauer, R.,Huber, R.,Lindberg, I.,Bode, W.,Than, M.E. (deposition date: 2003-05-07, release date: 2003-07-08, Last modification date: 2020-07-29)
Primary citationHenrich, S.,Cameron, A.,Bourenkov, G.P.,Kiefersauer, R.,Huber, R.,Lindberg, I.,Bode, W.,Than, M.E.
The Crystal Structure of the Proprotein Processing Proteinase Furin Explains its Stringent Specificity
Nat.Struct.Biol., 10:520-526, 2003
Cited by
PubMed: 12794637
DOI: 10.1038/nsb941
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

217705

数据于2024-03-27公开中

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