1GAR
TOWARDS STRUCTURE-BASED DRUG DESIGN: CRYSTAL STRUCTURE OF A MULTISUBSTRATE ADDUCT COMPLEX OF GLYCINAMIDE RIBONUCLEOTIDE TRANSFORMYLASE AT 1.96 ANGSTROMS RESOLUTION
Summary for 1GAR
Entry DOI | 10.2210/pdb1gar/pdb |
Descriptor | GLYCINAMIDE RIBONUCLEOTIDE TRANSFORMYLASE, N-[4-[[3-(2,4-DIAMINO-1,6-DIHYDRO-6-OXO-4-PYRIMIDINYL)-PROPYL]-[2-((2-OXO-2-((4-PHOSPHORIBOXY)-BUTYL)-AMINO)-ETHYL)-THIO-ACETYL]-AMINO]BENZOYL]-1-GLUTAMIC ACID (3 entities in total) |
Functional Keywords | transferase (formyl) |
Biological source | Escherichia coli |
Total number of polymer chains | 2 |
Total formula weight | 47963.85 |
Authors | Wilson, I.A.,Klein, C.,Chen, P.,Arevalo, J.H. (deposition date: 1994-12-08, release date: 1995-07-10, Last modification date: 2024-02-07) |
Primary citation | Klein, C.,Chen, P.,Arevalo, J.H.,Stura, E.A.,Marolewski, A.,Warren, M.S.,Benkovic, S.J.,Wilson, I.A. Towards structure-based drug design: crystal structure of a multisubstrate adduct complex of glycinamide ribonucleotide transformylase at 1.96 A resolution. J.Mol.Biol., 249:153-175, 1995 Cited by PubMed: 7776369DOI: 10.1006/jmbi.1995.0286 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.96 Å) |
Structure validation
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