1FQ7
X-RAY STRUCTURE OF INHIBITOR CP-72,647 BOUND TO SACCHAROPEPSIN
1FQ7 の概要
エントリーDOI | 10.2210/pdb1fq7/pdb |
関連するPDBエントリー | 1dp5 1fq4 1fq5 1fq6 1fq8 2jxr |
関連するBIRD辞書のPRD_ID | PRD_000564 |
分子名称 | SACCHAROPEPSIN, beta-D-arabino-hexopyranos-2-ulose-(1-2)-beta-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, N-(tert-butoxycarbonyl)-L-phenylalanyl-N-[(2S,3S,5R)-1-cyclohexyl-3-hydroxy-7-methyl-5-(methylcarbamoyl)octan-2-yl]-L-histidinamide, ... (5 entities in total) |
機能のキーワード | hydrophobic inhibitor, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
由来する生物種 | Saccharomyces cerevisiae (baker's yeast) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 37587.46 |
構造登録者 | Cronin, N.B.,Badasso, M.O.,Tickle, I.J.,Dreyer, T.,Hoover, D.J.,Rosati, R.L.,Humblet, C.C.,Lunney, E.A.,Cooper, J.B. (登録日: 2000-09-04, 公開日: 2000-09-20, 最終更新日: 2020-07-29) |
主引用文献 | Cronin, N.B.,Badasso, M.O.,J Tickle, I.,Dreyer, T.,Hoover, D.J.,Rosati, R.L.,Humblet, C.C.,Lunney, E.A.,Cooper, J.B. X-ray structures of five renin inhibitors bound to saccharopepsin: exploration of active-site specificity. J.Mol.Biol., 303:745-760, 2000 Cited by PubMed: 11061973DOI: 10.1006/jmbi.2000.4181 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.8 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード