1EH4
BINARY COMPLEX OF CASEIN KINASE-1 FROM S. POMBE WITH AN ATP COMPETITIVE INHIBITOR, IC261
Summary for 1EH4
Entry DOI | 10.2210/pdb1eh4/pdb |
Related | 1CSN 2CSN |
Descriptor | CASEIN KINASE-1, SULFATE ION, 3-[(2,4,6-TRIMETHOXY-PHENYL)-METHYLENE]-INDOLIN-2-ONE, ... (4 entities in total) |
Functional Keywords | protein kinase, casein kinase-1, protein-inhibitor binary complex, transferase |
Biological source | Schizosaccharomyces pombe (fission yeast) |
Cellular location | Cytoplasm: P40233 |
Total number of polymer chains | 2 |
Total formula weight | 70433.83 |
Authors | Mashhoon, N.,Demaggio, A.J.,Tereshko, V.,Bergmeier, S.C.,Egli, M.,Hoekstra, M.F.,Kuret, J. (deposition date: 2000-02-18, release date: 2001-09-19, Last modification date: 2024-03-13) |
Primary citation | Mashhoon, N.,Demaggio, A.J.,Tereshko, V.,Bergmeier, S.C.,Egli, M.,Hoekstra, M.F.,Kuret, J. Crystal Structure of a Conformation-Selective Casein Kinase-1 Inhibitor J.Biol.Chem., 275:20052-20060, 2000 Cited by PubMed: 10749871DOI: 10.1074/jbc.M001713200 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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