1RT5
HIV-1 REVERSE TRANSCRIPTASE COMPLEXED WITH UC10
Summary for 1RT5
Entry DOI | 10.2210/pdb1rt5/pdb |
Descriptor | HIV-1 REVERSE TRANSCRIPTASE, PHOSPHATE ION, N-[4-CLORO-3-(T-BUTYLOXOME)PHENYL-2-METHYL-3-FURAN-CARBOTHIAMIDE, ... (5 entities in total) |
Functional Keywords | nucleotidyltransferase, hiv-1 reverse transcriptase, aids, nonnucleoside inhibition, drug design |
Biological source | HIV-1 M:B_HXB2R More |
Cellular location | Matrix protein p17: Virion (Potential). Capsid protein p24: Virion (Potential). Nucleocapsid protein p7: Virion (Potential). Reverse transcriptase/ribonuclease H: Virion (Potential). Integrase: Virion (Potential): P04585 P04585 |
Total number of polymer chains | 2 |
Total formula weight | 116439.83 |
Authors | Ren, J.,Stammers, D.K.,Stuart, D.I. (deposition date: 1998-07-29, release date: 1999-07-29, Last modification date: 2023-08-09) |
Primary citation | Ren, J.,Esnouf, R.M.,Hopkins, A.L.,Warren, J.,Balzarini, J.,Stuart, D.I.,Stammers, D.K. Crystal structures of HIV-1 reverse transcriptase in complex with carboxanilide derivatives. Biochemistry, 37:14394-14403, 1998 Cited by PubMed: 9772165DOI: 10.1021/bi981309m PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.9 Å) |
Structure validation
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