1GZL
Crystal structure of C14linkmid/IQN17: a cross-linked inhibitor of HIV-1 entry bound to the gp41 hydrophobic pocket
Summary for 1GZL
Entry DOI | 10.2210/pdb1gzl/pdb |
Related | 1DGC 1E7T 1ENV 1FAV 1GCL 1GCM 1GK6 1IHQ 1IJ0 1IJ1 1IJ2 1IJ3 1KQL 1PIQ 1SWI 1TMZ 1YSA 1ZII 1ZIJ 1ZIK 1ZIL 1ZIM 1ZTA 2DGC 2ZTA |
Descriptor | FUSION PROTEIN BETWEEN THE HYDROPHOBIC POCKET OF HIV GP41 AND GENERAL CONTROL PROTEIN GCN4-PIQI, ENVELOPE GLYCOPROTEIN GP41, CHLORIDE ION, ... (5 entities in total) |
Functional Keywords | glycoprotein, hiv entry, inhibitor, cross-link, gp41, coiled coil |
Biological source | SACCHAROMYCES CEREVISIAE (BAKER'S YEAST) More |
Total number of polymer chains | 4 |
Total formula weight | 14553.81 |
Authors | Sia, S.K.,Carr, P.A.,Cochran, A.G.,Malashkevich, V.M.,Kim, P.S. (deposition date: 2002-05-23, release date: 2002-10-10, Last modification date: 2024-10-16) |
Primary citation | Sia, S.K.,Carr, P.A.,Cochran, A.G.,Malashkevich, V.M.,Kim, P.S. Short Constrained Peptides that Inhibit HIV-1 Entry Proc.Natl.Acad.Sci.USA, 99:14664-, 2002 Cited by PubMed: 12417739DOI: 10.1073/PNAS.232566599 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
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