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1BKF

FK506 BINDING PROTEIN FKBP MUTANT R42K/H87V COMPLEX WITH IMMUNOSUPPRESSANT FK506

Summary for 1BKF
Entry DOI10.2210/pdb1bkf/pdb
DescriptorFK506 BINDING PROTEIN, 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN (3 entities in total)
Functional Keywordsisomerase, rotamase
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm, cytosol : P62942
Total number of polymer chains1
Total formula weight12573.50
Authors
Itoh, S.,Decenzo, M.T.,Livingston, D.J.,Pearlman, D.A.,Navia, M.A. (deposition date: 1995-10-18, release date: 1996-08-01, Last modification date: 2024-02-07)
Primary citationItoh, S.,Decenzo, M.T.,Livingston, D.J.,Pearlman, D.A.,Navia, M.A.
Conformation of Fk506 in X-Ray Structures of its Complexes with Human Recombinant Fkbp12 Mutants
Bioorg.Med.Chem.Lett., 5:1983-, 1995
Cited by
Experimental method
X-RAY DIFFRACTION (1.6 Å)
Structure validation

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