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10NL

Xenopus KCNQ1 in complex with UCL2077

This is a non-PDB format compatible entry.
Summary for 10NL
Entry DOI10.2210/pdb10nl/pdb
EMDB information75306
DescriptorCalmodulin-1, Potassium voltage-gated channel subfamily KQT member 1, 1,1,1-triphenyl-N-[(pyridin-3-yl)methyl]methanamine (3 entities in total)
Functional Keywordspotassium ion channel protein, transport protein
Biological sourceHomo sapiens (human)
More
Total number of polymer chains8
Total formula weight317611.64
Authors
Kyriakis, E.,Eldstrom, J.,Van Petegem, F.,Fedida, D. (deposition date: 2026-01-28, release date: 2026-09-02)
Primary citationKyriakis, E.,Roscioni, A.,Eldstrom, J.,Sastre, D.,Dou, Y.,Taddei, A.,Molinarolo, S.,Tian, M.,Maragliano, L.,Van Petegem, F.,Fedida, D.
Structural and kinetic mechanisms of state-dependent potassium channel inhibition
Sci Adv, 2026
Experimental method
ELECTRON MICROSCOPY (3.81 Å)
Structure validation

259015

PDB entries from 2026-09-02

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