Entity
| Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
| 1 | A (A) | Mast/stem cell growth factor receptor | polymer | 359 | 41163.3 | 1 | UniProt (A0A0U2N547) | Homo sapiens (human) | |
| 2 | B (A) | (4R)-2-METHYLPENTANE-2,4-DIOL | non-polymer | 118.2 | 1 | Chemie (MRD) PubChem (7870) PubChem (5288834) PubChem (5288845) | |||
| 3 | C (A) | N~2~-methyl-N~4~-{(5P)-5-(1-methyl-1H-pyrazol-4-yl)-4-[(propan-2-yl)oxy]pyridin-2-yl}pyrimidine-2,4-diamine | non-polymer | 339.4 | 1 | Chemie (A1CZZ) | |||
| 4 | D (A) | water | water | 18.0 | 488 | Chemie (HOH) |
Sequence modifications
A: 544 - 935 (UniProt: A0A0U2N547)
| PDB | External Database | Details |
|---|---|---|
| Met 519 | - | initiating methionine |
| Ser 520 | - | expression tag |
| Tyr 521 | - | expression tag |
| Tyr 522 | - | expression tag |
| His 523 | - | expression tag |
| His 524 | - | expression tag |
| His 525 | - | expression tag |
| His 526 | - | expression tag |
| His 527 | - | expression tag |
| His 528 | - | expression tag |
| Asp 529 | - | expression tag |
| Tyr 530 | - | expression tag |
| Asp 531 | - | expression tag |
| Ile 532 | - | expression tag |
| Pro 533 | - | expression tag |
| Thr 534 | - | expression tag |
| Thr 535 | - | expression tag |
| Glu 536 | - | expression tag |
| Asn 537 | - | expression tag |
| Leu 538 | - | expression tag |
| Tyr 539 | - | expression tag |
| Phe 540 | - | expression tag |
| Gln 541 | - | expression tag |
| Gly 542 | - | expression tag |
| Pro 543 | - | expression tag |
| Ala 654 | Val 650 | engineered mutation |
| - | Gln 690 | deletion |
| - | Glu 691 | deletion |
| - | Asp 692 | deletion |
| - | His 693 | deletion |
| - | Ala 694 | deletion |
| - | Glu 695 | deletion |
| - | Ala 696 | deletion |
| - | Ala 697 | deletion |
| - | Leu 698 | deletion |
| - | Tyr 699 | deletion |
| - | Lys 700 | deletion |
| - | Asn 701 | deletion |
| - | Leu 702 | deletion |
| - | Leu 703 | deletion |
| - | His 704 | deletion |
| - | Ser 705 | deletion |
| - | Lys 706 | deletion |
| - | Glu 707 | deletion |
| - | Ser 708 | deletion |
| - | Ser 709 | deletion |
| - | Cys 710 | deletion |
| - | Asp 711 | deletion |
| - | Ser 712 | deletion |
| - | Thr 713 | deletion |
| - | Asn 714 | deletion |
| - | Glu 715 | deletion |
| - | Tyr 716 | deletion |
| - | Met 717 | deletion |
| - | Asp 718 | deletion |
| - | Met 719 | deletion |
| - | Lys 720 | deletion |
| - | Pro 721 | deletion |
| - | Gly 722 | deletion |
| - | Val 723 | deletion |
| - | Ser 724 | deletion |
| - | Tyr 725 | deletion |
| - | Val 726 | deletion |
| - | Val 727 | deletion |
| - | Pro 728 | deletion |
| - | Thr 729 | deletion |
| - | Lys 730 | deletion |
| - | Ala 731 | deletion |
| - | Asp 732 | deletion |
| - | Lys 733 | deletion |
| - | Arg 734 | deletion |
| - | Arg 735 | deletion |
| - | Ser 736 | deletion |
| - | Val 737 | deletion |
| - | Arg 738 | deletion |
| - | Ile 739 | deletion |
| - | Gly 740 | deletion |
| - | Ser 741 | deletion |
| - | Tyr 742 | deletion |
| - | Ile 743 | deletion |
| - | Glu 744 | deletion |
| - | Arg 745 | deletion |
| - | Asp 746 | deletion |
| Thr 752 | Val 747 | conflict |
| Ser 753 | Thr 748 | conflict |
Sequence viewer
Contents of the asymmetric unit
| Polymers | Number of chains | 1 |
| Total formula weight | 41163.3 | |
| Non-Polymers* | Number of molecules | 2 |
| Total formula weight | 457.6 | |
| All* | Total formula weight | 41620.9 |






