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9Z1L

Structure of KIT V654A mutant with Compound 1

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
Mast/stem cell growth factor receptorpolymer35941163.31UniProt (A0A0U2N547)Homo sapiens (human)
2B
(A)
(4R)-2-METHYLPENTANE-2,4-DIOLnon-polymer118.21Chemie (MRD)
PubChem (7870)
PubChem (5288834)
PubChem (5288845)
3C
(A)
N~2~-methyl-N~4~-{(5P)-5-(1-methyl-1H-pyrazol-4-yl)-4-[(propan-2-yl)oxy]pyridin-2-yl}pyrimidine-2,4-diaminenon-polymer339.41Chemie (A1CZZ)
4D
(A)
waterwater18.0488Chemie (HOH)
Sequence modifications
A: 544 - 935 (UniProt: A0A0U2N547)
PDBExternal DatabaseDetails
Met 519-initiating methionine
Ser 520-expression tag
Tyr 521-expression tag
Tyr 522-expression tag
His 523-expression tag
His 524-expression tag
His 525-expression tag
His 526-expression tag
His 527-expression tag
His 528-expression tag
Asp 529-expression tag
Tyr 530-expression tag
Asp 531-expression tag
Ile 532-expression tag
Pro 533-expression tag
Thr 534-expression tag
Thr 535-expression tag
Glu 536-expression tag
Asn 537-expression tag
Leu 538-expression tag
Tyr 539-expression tag
Phe 540-expression tag
Gln 541-expression tag
Gly 542-expression tag
Pro 543-expression tag
Ala 654Val 650engineered mutation
-Gln 690deletion
-Glu 691deletion
-Asp 692deletion
-His 693deletion
-Ala 694deletion
-Glu 695deletion
-Ala 696deletion
-Ala 697deletion
-Leu 698deletion
-Tyr 699deletion
-Lys 700deletion
-Asn 701deletion
-Leu 702deletion
-Leu 703deletion
-His 704deletion
-Ser 705deletion
-Lys 706deletion
-Glu 707deletion
-Ser 708deletion
-Ser 709deletion
-Cys 710deletion
-Asp 711deletion
-Ser 712deletion
-Thr 713deletion
-Asn 714deletion
-Glu 715deletion
-Tyr 716deletion
-Met 717deletion
-Asp 718deletion
-Met 719deletion
-Lys 720deletion
-Pro 721deletion
-Gly 722deletion
-Val 723deletion
-Ser 724deletion
-Tyr 725deletion
-Val 726deletion
-Val 727deletion
-Pro 728deletion
-Thr 729deletion
-Lys 730deletion
-Ala 731deletion
-Asp 732deletion
-Lys 733deletion
-Arg 734deletion
-Arg 735deletion
-Ser 736deletion
-Val 737deletion
-Arg 738deletion
-Ile 739deletion
-Gly 740deletion
-Ser 741deletion
-Tyr 742deletion
-Ile 743deletion
-Glu 744deletion
-Arg 745deletion
-Asp 746deletion
Thr 752Val 747conflict
Ser 753Thr 748conflict
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight41163.3
Non-Polymers*Number of molecules2
Total formula weight457.6
All*Total formula weight41620.9
*Water molecules are not included.

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PDB entries from 2026-04-01

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