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9DC6

Structure of J-PKAc chimera in complex with Aplithianine e1

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B
(A, B)
cAMP-dependent protein kinase catalytic subunit alphapolymer40547512.02UniProt (P17612)Homo sapiens (human)PKA C-alpha
2C, D
(I, J)
cAMP-dependent protein kinase inhibitor alphapolymer202226.42UniProt (P61925)Homo sapiensPKI-alpha,cAMP-dependent protein kinase inhibitor,muscle/brain isoform
3E, F
(A, B)
N-(2-aminoethyl)-4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-3,4-dihydro-2H-1,4-thiazine-6-carboxamidenon-polymer304.42Chemie (A1A3I)
Sequence modifications
A, B: 70 - 405 (UniProt: P17612)
PDBExternal DatabaseDetails
Gly 1-expression tag
Lys 2-expression tag
Asp 3-expression tag
Tyr 4-expression tag
Tyr 5-expression tag
Gln 6-expression tag
Thr 7-expression tag
Leu 8-expression tag
Gly 9-expression tag
Leu 10-expression tag
Ala 11-expression tag
Arg 12-expression tag
Gly 13-expression tag
Ala 14-expression tag
Ser 15-expression tag
Asp 16-expression tag
Glu 17-expression tag
Glu 18-expression tag
Ile 19-expression tag
Lys 20-expression tag
Arg 21-expression tag
Ala 22-expression tag
Tyr 23-expression tag
Arg 24-expression tag
Arg 25-expression tag
Gln 26-expression tag
Ala 27-expression tag
Leu 28-expression tag
Arg 29-expression tag
Tyr 30-expression tag
His 31-expression tag
Pro 32-expression tag
Asp 33-expression tag
Lys 34-expression tag
Asn 35-expression tag
Lys 36-expression tag
Glu 37-expression tag
Pro 38-expression tag
Gly 39-expression tag
Ala 40-expression tag
Glu 41-expression tag
Glu 42-expression tag
Lys 43-expression tag
Phe 44-expression tag
Lys 45-expression tag
Glu 46-expression tag
Ile 47-expression tag
Ala 48-expression tag
Glu 49-expression tag
Ala 50-expression tag
Tyr 51-expression tag
Asp 52-expression tag
Val 53-expression tag
Leu 54-expression tag
Ser 55-expression tag
Asp 56-expression tag
Pro 57-expression tag
Arg 58-expression tag
Lys 59-expression tag
Arg 60-expression tag
Glu 61-expression tag
Ile 62-expression tag
Phe 63-expression tag
Asp 64-expression tag
Arg 65-expression tag
Tyr 66-expression tag
Gly 67-expression tag
Glu 68-expression tag
Glu 69-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight99476.8
Non-Polymers*Number of molecules2
Total formula weight608.7
All*Total formula weight100085.5
*Water molecules are not included.

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PDB entries from 2025-07-09

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