8PJK
ST171-bound serotonin 5-HT1A receptor - Gi Protein Complex
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Guanine nucleotide-binding protein G(i) subunit alpha-1 | polymer | 354 | 40414.0 | 1 | UniProt (P63096) Pfam (PF00503) In PDB | Homo sapiens (human) | |
2 | B | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 | polymer | 352 | 38810.4 | 1 | UniProt (P62873) Pfam (PF00400) In PDB | Homo sapiens (human) | |
3 | G | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 | polymer | 71 | 7861.1 | 1 | UniProt (P59768) Pfam (PF00631) In PDB | Homo sapiens (human) | G gamma-I |
4 | R | 5-hydroxytryptamine receptor 1A | polymer | 466 | 51431.6 | 1 | UniProt (P08908) Pfam (PF00001) In PDB | Homo sapiens (human) | 5-HT-1A,5-HT1A,G-21,Serotonin receptor 1A |
5 | R | CHOLESTEROL | non-polymer | 386.7 | 2 | Chemie (CLR) | |||
6 | R | 6-[3-[2-(2-methoxyphenoxy)ethylamino]propoxy]-4~{H}-1,4-benzoxazin-3-one | non-polymer | 372.4 | 1 | Chemie (ZL9) | |||
7 | R | (2R)-1-(heptadecanoyloxy)-3-{[(R)-hydroxy{[(1R,2R,3R,4R,5S,6R)-2,3,5,6-tetrahydroxy-4-(phosphonooxy)cyclohexyl]oxy}phosphoryl]oxy}propan-2-yl (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate | non-polymer | 953.1 | 1 | Chemie (T7M) | |||
8 | water | water | 18.0 | 39 | Chemie (HOH) |
Sequence modifications
A: 1 - 354 (UniProt: P63096)
B: 2 - 340 (UniProt: P62873)
R: 1 - 422 (UniProt: P08908)
PDB | External Database | Details |
---|---|---|
Asn 47 | Ser 47 | conflict |
Ala 203 | Gly 203 | conflict |
Ala 245 | Glu 245 | conflict |
Ser 326 | Ala 326 | conflict |
PDB | External Database | Details |
---|---|---|
Met -11 | - | initiating methionine |
His -10 | - | expression tag |
His -9 | - | expression tag |
His -8 | - | expression tag |
His -7 | - | expression tag |
His -6 | - | expression tag |
His -5 | - | expression tag |
His -4 | - | expression tag |
His -3 | - | expression tag |
Gly -2 | - | expression tag |
Ser -1 | - | expression tag |
Ser 0 | - | expression tag |
Gly 1 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Met -43 | - | initiating methionine |
Lys -42 | - | expression tag |
Thr -41 | - | expression tag |
Ile -40 | - | expression tag |
Ile -39 | - | expression tag |
Ala -38 | - | expression tag |
Leu -37 | - | expression tag |
Ser -36 | - | expression tag |
Tyr -35 | - | expression tag |
Ile -34 | - | expression tag |
Phe -33 | - | expression tag |
Cys -32 | - | expression tag |
Leu -31 | - | expression tag |
Val -30 | - | expression tag |
Phe -29 | - | expression tag |
Ala -28 | - | expression tag |
Asp -27 | - | expression tag |
Tyr -26 | - | expression tag |
Lys -25 | - | expression tag |
Asp -24 | - | expression tag |
Asp -23 | - | expression tag |
Asp -22 | - | expression tag |
Asp -21 | - | expression tag |
Ala -20 | - | expression tag |
Ala -19 | - | expression tag |
Ala -18 | - | expression tag |
Ala -17 | - | expression tag |
His -16 | - | expression tag |
His -15 | - | expression tag |
His -14 | - | expression tag |
His -13 | - | expression tag |
His -12 | - | expression tag |
His -11 | - | expression tag |
His -10 | - | expression tag |
His -9 | - | expression tag |
His -8 | - | expression tag |
His -7 | - | expression tag |
Glu -6 | - | expression tag |
Asn -5 | - | expression tag |
Leu -4 | - | expression tag |
Tyr -3 | - | expression tag |
Phe -2 | - | expression tag |
Gln -1 | - | expression tag |
Gly 0 | - | expression tag |
Trp 125 | Leu 125 | conflict |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 138517.1 | |
Non-Polymers* | Number of molecules | 4 |
Total formula weight | 2098.8 | |
All* | Total formula weight | 140615.9 |