Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

8FGZ

Crystal structure of mutant Androgen Receptor ligand binding domain L702H/H875Y/F877L with DHT

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
Androgen receptorpolymer25830110.21UniProt (P10275)
Pfam (PF00104)
Homo sapiens (human)Dihydrotestosterone receptor,Nuclear receptor subfamily 3 group C member 4
2B
(A)
5-ALPHA-DIHYDROTESTOSTERONEnon-polymer290.41Chemie (DHT)
PubChem (16395945)
PubChem (1779160)
PubChem (23729584)
PubChem (44264584)
PubChem (44307156)
PubChem (44308180)
PubChem (44314545)
PubChem (1779165)
PubChem (1779163)
PubChem (44403751)
PubChem (54132599)
PubChem (57253355)
PubChem (2748143)
PubChem (11302)
PubChem (968803)
PubChem (6951009)
PubChem (124916763)
PubChem (67080676)
PubChem (68213431)
PubChem (70627790)
PubChem (133612463)
PubChem (11869360)
PubChem (15)
PubChem (76333143)
PubChem (10635)
PubChem (90350225)
PubChem (147320)
PubChem (16111632)
PubChem (667503)
PubChem (928651)
PubChem (124305346)
PubChem (124335861)
PubChem (124350819)
PubChem (124362930)
PubChem (124402106)
PubChem (124420348)
PubChem (124907326)
PubChem (124907327)
PubChem (6432518)
PubChem (7052570)
PubChem (7052571)
PubChem (9965809)
PubChem (134753818)
PubChem (10379482)
PubChem (10902374)
PubChem (11860392)
PubChem (11867857)
PubChem (11867858)
PubChem (11867859)
PubChem (11867860)
PubChem (11869358)
PubChem (11869359)
PubChem (11869361)
PubChem (11914201)
PubChem (11920866)
PubChem (139564330)
PubChem (141909893)
PubChem (142776876)
PubChem (145087815)
PubChem (12446746)
PubChem (12446747)
PubChem (12446748)
PubChem (12446749)
PubChem (12446752)
PubChem (156740897)
PubChem (162854571)
PubChem (162854572)
PubChem (162854573)
PubChem (164663566)
PubChem (165146196)
PubChem (165431280)
3C, D
(A)
SULFATE IONnon-polymer96.12Chemie (SO4)
4E
(A)
waterwater18.077Chemie (HOH)
Sequence modifications
A: 663 - 920 (UniProt: P10275)
PDBExternal DatabaseDetails
His 702Leu 702engineered mutation
Tyr 875His 875engineered mutation
Leu 877Phe 877engineered mutation
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight30110.2
Non-Polymers*Number of molecules3
Total formula weight482.6
All*Total formula weight30592.7
*Water molecules are not included.

251174

PDB entries from 2026-03-25

PDB statisticsPDBj update infoContact PDBjnumon