8BX6
Crystal structure of JAK2 JH1 in complex with cerdulatinib
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Tyrosine-protein kinase JAK2 | polymer | 316 | 37268.3 | 1 | UniProt (O60674) Pfam (PF07714) In PDB | Homo sapiens (human) | Janus kinase 2,JAK-2 |
2 | A | Cerdulatinib | non-polymer | 445.5 | 1 | Chemie (S5I) | |||
3 | water | water | 18.0 | 231 | Chemie (HOH) |
Sequence modifications
A: 840 - 1132 (UniProt: O60674)
PDB | External Database | Details |
---|---|---|
Met 817 | - | initiating methionine |
His 818 | - | expression tag |
His 819 | - | expression tag |
His 820 | - | expression tag |
His 821 | - | expression tag |
His 822 | - | expression tag |
His 823 | - | expression tag |
Ser 824 | - | expression tag |
Ser 825 | - | expression tag |
Gly 826 | - | expression tag |
Val 827 | - | expression tag |
Asp 828 | - | expression tag |
Leu 829 | - | expression tag |
Gly 830 | - | expression tag |
Thr 831 | - | expression tag |
Glu 832 | - | expression tag |
Asn 833 | - | expression tag |
Leu 834 | - | expression tag |
Tyr 835 | - | expression tag |
Phe 836 | - | expression tag |
Gln 837 | - | expression tag |
Ser 838 | - | expression tag |
Met 839 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 37268.3 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 445.5 | |
All* | Total formula weight | 37713.8 |