8AYL
Resting state GluA1/A2 AMPA receptor in complex with TARP gamma 8 and ligand JNJ-61432059
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | B, D | Isoform Flip of Glutamate receptor 2 | polymer | 860 | 96247.1 | 2 | UniProt (P19491) Pfam (PF01094) Pfam (PF10613) Pfam (PF00060) In PDB | Rattus norvegicus (Norway rat) | GluR-2,AMPA-selective glutamate receptor 2,GluR-B,GluR-K2,Glutamate receptor ionotropic,AMPA 2,GluA2 |
2 | J, I | Voltage-dependent calcium channel gamma-8 subunit | polymer | 423 | 43576.0 | 2 | UniProt (Q8VHW5) Pfam (PF00822) In PDB | Rattus norvegicus (Norway rat) | Neuronal voltage-gated calcium channel gamma-8 subunit,Transmembrane AMPAR regulatory protein gamma-8,TARP gamma-8 |
3 | A, C | Isoform Flip of Glutamate receptor 1 | polymer | 915 | 102661.9 | 2 | UniProt (P19490) Pfam (PF01094) Pfam (PF10613) Pfam (PF00060) In PDB | Rattus norvegicus (Norway rat) | GluR-1,AMPA-selective glutamate receptor 1,GluR-A,GluR-K1,Glutamate receptor ionotropic,AMPA 1,GluA1 |
4 | B, A, D, C | {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid | non-polymer | 409.3 | 4 | Chemie (ZK1) | |||
5 | C, B, A, D | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate | non-polymer | 356.5 | 4 | Chemie (OLC) | |||
6 | C, B, A, D | PALMITIC ACID | non-polymer | 256.4 | 8 | Chemie (PLM) | |||
7 | C, B, J, I, A... | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate | non-polymer | 760.1 | 6 | Chemie (POV) | |||
8 | J, I | 5-[2-(4-fluorophenyl)-7-(4-oxidanylpiperidin-1-yl)pyrazolo[1,5-c]pyrimidin-3-yl]-1,3-dihydroindol-2-one | non-polymer | 443.5 | 2 | Chemie (OIJ) |
Sequence modifications
B, D: -20 - 839 (UniProt: P19491)
J, I: 2 - 417 (UniProt: Q8VHW5)
A, C: -25 - 889 (UniProt: P19490)
PDB | External Database | Details |
---|---|---|
Arg 586 | Gln 607 | variant |
PDB | External Database | Details |
---|---|---|
Gly 1 | - | expression tag |
Leu 418 | - | expression tag |
Glu 419 | - | expression tag |
Val 420 | - | expression tag |
Leu 421 | - | expression tag |
Phe 422 | - | expression tag |
Gln 423 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Asp -6 | - | insertion |
Tyr -5 | - | insertion |
Lys -4 | - | insertion |
Asp -3 | - | insertion |
Asp -2 | - | insertion |
Asp -1 | - | insertion |
Asp 0 | - | insertion |
Lys 1 | - | insertion |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 6 |
Total formula weight | 484970.0 | |
Non-Polymers* | Number of molecules | 24 |
Total formula weight | 10562.0 | |
All* | Total formula weight | 495531.9 |