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7ZV9

Crystal structure of FLT3 in complex with a monomeric FLT3 Ligand variant

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, C, E, G, I...Fms-related tyrosine kinase 3 ligandpolymer15517764.28UniProt (P49771)
Pfam (PF02947)
In PDB
Homo sapiens (human)Flt3 ligand,Flt3L,SL cytokine
2B, D, F, H, J...Receptor-type tyrosine-protein kinase FLT3polymer58265307.88UniProt (P36888)
Pfam (PF00047)
In PDB
Homo sapiens (human)FL cytokine receptor,Fetal liver kinase-2,FLK-2,Fms-like tyrosine kinase 3,FLT-3,Stem cell tyrosine kinase 1,STK-1
3Q, R, S, T, U...2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranosebranched424.46In PDB
GlyTouCan (G42666HT)
4B, H, P2-acetamido-2-deoxy-beta-D-glucopyranosenon-polymer221.24Chemie (NAG)
Sequence modifications
A, C, E, G, I, K, M, O: 1 - 134 (UniProt: P49771)
PDBExternal DatabaseDetails
Met -20-initiating methionine
Gly -19-expression tag
Ser -18-expression tag
Ser -17-expression tag
His -16-expression tag
His -15-expression tag
His -14-expression tag
His -13-expression tag
His -12-expression tag
His -11-expression tag
Ser -10-expression tag
Ser -9-expression tag
Gly -8-expression tag
Leu -7-expression tag
Val -6-expression tag
Pro -5-expression tag
Arg -4-expression tag
Gly -3-expression tag
Ser -2-expression tag
His -1-expression tag
Met 0-expression tag
Asp 27Leu 53engineered mutation
B, D, F, H, J, L, N, P: 1 - 541 (UniProt: P36888)
PDBExternal DatabaseDetails
Met 227Thr 227conflict
Gly 542-expression tag
Ser 543-expression tag
Ser 544-expression tag
Gly 545-expression tag
Leu 546-expression tag
Val 547-expression tag
Pro 548-expression tag
Arg 549-expression tag
Gly 550-expression tag
Ser 551-expression tag
Gly 552-expression tag
Gly 553-expression tag
Ser 554-expression tag
Gly 555-expression tag
Gly 556-expression tag
Ser 557-expression tag
Gly 558-expression tag
Leu 559-expression tag
Asn 560-expression tag
Asp 561-expression tag
Ile 562-expression tag
Phe 563-expression tag
Glu 564-expression tag
Ala 565-expression tag
Gln 566-expression tag
Lys 567-expression tag
Ile 568-expression tag
Glu 569-expression tag
Trp 570-expression tag
His 571-expression tag
Glu 572-expression tag
Gly 573-expression tag
Arg 574-expression tag
Thr 575-expression tag
Lys 576-expression tag
His 577-expression tag
His 578-expression tag
His 579-expression tag
His 580-expression tag
His 581-expression tag
His 582-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains16
Total formula weight664576.5
BranchedNumber of molecules6
Total formula weight2546.4
Non-Polymers*Number of molecules4
Total formula weight884.8
All*Total formula weight668007.8
*Water molecules are not included.

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PDB entries from 2024-06-12

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