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7ZU2

Crystal structure of mutant AR-LBD (Q799E) bound to dihydrotestosterone

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
Androgen receptorpolymer24929047.11UniProt (P10275)
Pfam (PF00104)
Homo sapiens (human)Dihydrotestosterone receptor,Nuclear receptor subfamily 3 group C member 4
2B
(A)
5-ALPHA-DIHYDROTESTOSTERONEnon-polymer290.41Chemie (DHT)
PubChem (16395945)
PubChem (1779160)
PubChem (15)
PubChem (10635)
PubChem (147320)
PubChem (23729584)
PubChem (44264584)
PubChem (44307156)
PubChem (44308180)
PubChem (44314545)
PubChem (1779165)
PubChem (1779163)
PubChem (44403751)
PubChem (667503)
PubChem (928651)
PubChem (54132599)
PubChem (57253355)
PubChem (67080676)
PubChem (2748143)
PubChem (68213431)
PubChem (70627790)
PubChem (76333143)
PubChem (6432518)
PubChem (11302)
PubChem (7052570)
PubChem (7052571)
PubChem (90350225)
PubChem (9965809)
PubChem (10379482)
PubChem (10902374)
PubChem (968803)
PubChem (11860392)
PubChem (11867857)
PubChem (11867858)
PubChem (11867859)
PubChem (11867860)
PubChem (11869358)
PubChem (11869359)
PubChem (11869361)
PubChem (11914201)
PubChem (11920866)
PubChem (12446746)
PubChem (12446747)
PubChem (12446748)
PubChem (12446749)
PubChem (12446752)
PubChem (6951009)
PubChem (124916763)
PubChem (133612463)
PubChem (11869360)
PubChem (124305346)
PubChem (124335861)
PubChem (124350819)
PubChem (124362930)
PubChem (124402106)
PubChem (124420348)
PubChem (124907326)
PubChem (124907327)
PubChem (16111632)
PubChem (134753818)
PubChem (139564330)
PubChem (141909893)
PubChem (142776876)
PubChem (145087815)
PubChem (156740897)
PubChem (162854571)
PubChem (162854572)
PubChem (162854573)
PubChem (164663566)
PubChem (165146196)
PubChem (165431280)
3C, D
(A)
IMIDAZOLEnon-polymer69.12Chemie (IMD)
4E
(A)
waterwater18.064Chemie (HOH)
Sequence modifications
A: 672 - 920 (UniProt: P10275)
PDBExternal DatabaseDetails
Glu 799Gln 799engineered mutation
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight29047.1
Non-Polymers*Number of molecules3
Total formula weight428.6
All*Total formula weight29475.7
*Water molecules are not included.

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PDB entries from 2026-04-01

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