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7RJ7

CRYSTAL STRUCTURE OF AP2 ASSOCIATED KINASE 1 ISOFORM 1 COMPLEXED WITH LIGAND 2-(1-AMINO-3-METHYLBUTYL)-6- (PYRIDIN-4-YL)QUINOLINE-4-CARBONITRILE

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, BAP2-associated protein kinase 1polymer31835978.22UniProt (Q3UHJ0)
Pfam (PF00069)
In PDB
Mus musculus (Mouse)Adaptor-associated kinase 1
2A, B2-[(1S)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrilenon-polymer316.42Chemie (5P6)
3BSULFATE IONnon-polymer96.16Chemie (SO4)
4waterwater18.0217Chemie (HOH)
Sequence modifications
A, B: 26 - 330 (UniProt: Q3UHJ0)
PDBExternal DatabaseDetails
Met 13-initiating methionine
His 14-expression tag
His 15-expression tag
His 16-expression tag
His 17-expression tag
His 18-expression tag
His 19-expression tag
Leu 20-expression tag
Val 21-expression tag
Pro 22-expression tag
Arg 23-expression tag
Gly 24-expression tag
Ser 25-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight71956.4
Non-Polymers*Number of molecules8
Total formula weight1209.2
All*Total formula weight73165.6
*Water molecules are not included.

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PDB entries from 2024-06-12

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