7F8U
Crystal structure of the cholecystokinin receptor CCKAR in complex with lintitript
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Fusion protein of Cholecystokinin receptor type A and Endolysin | polymer | 534 | 60450.4 | 1 | UniProt (P32238) UniProt (P00720) Pfam (PF00001) Pfam (PF00959) In PDB | Homo sapiens (Human) | CCK-A receptor,CCK-AR,Cholecystokinin-1 receptor,CCK1-R,Lysis protein,Lysozyme,Muramidase |
2 | A | 2-[2-[[4-(2-chlorophenyl)-1,3-thiazol-2-yl]carbamoyl]indol-1-yl]ethanoic acid | non-polymer | 411.9 | 1 | Chemie (1OE) |
Sequence modifications
A: 37 - 240 (UniProt: P32238)
A: 1241 - 1400 (UniProt: P00720)
A: 302 - 375 (UniProt: P32238)
PDB | External Database | Details |
---|---|---|
Asp -8 | - | expression tag |
Tyr -7 | - | expression tag |
Lys -6 | - | expression tag |
Asp -5 | - | expression tag |
Asp -4 | - | expression tag |
Asp -3 | - | expression tag |
Asp -2 | - | expression tag |
Gly -1 | - | expression tag |
Ala 0 | - | expression tag |
Pro 1 | - | expression tag |
Asp 2 | - | expression tag |
Val 3 | - | expression tag |
Val 4 | - | expression tag |
Asp 5 | - | expression tag |
Ser 6 | - | expression tag |
Leu 7 | - | expression tag |
Leu 8 | - | expression tag |
Val 9 | - | expression tag |
Asn 10 | - | expression tag |
Gly 11 | - | expression tag |
Ser 12 | - | expression tag |
Asn 13 | - | expression tag |
Ile 14 | - | expression tag |
Thr 15 | - | expression tag |
Pro 16 | - | expression tag |
Pro 17 | - | expression tag |
Cys 18 | - | expression tag |
Glu 19 | - | expression tag |
Leu 20 | - | expression tag |
Gly 21 | - | expression tag |
Leu 22 | - | expression tag |
Glu 23 | - | expression tag |
Asn 24 | - | expression tag |
Glu 25 | - | expression tag |
Thr 26 | - | expression tag |
Leu 27 | - | expression tag |
Phe 28 | - | expression tag |
Cys 29 | - | expression tag |
Leu 30 | - | expression tag |
Asp 31 | - | expression tag |
Gln 32 | - | expression tag |
Pro 33 | - | expression tag |
Arg 34 | - | expression tag |
Pro 35 | - | expression tag |
Ser 36 | - | expression tag |
Asn 87 | Asp 87 | conflict |
Trp 130 | Phe 130 | conflict |
PDB | External Database | Details |
---|---|---|
Gly 1251 | Arg 12 | conflict |
Thr 1293 | Cys 54 | conflict |
Ala 1336 | Cys 97 | conflict |
Arg 1376 | Ile 137 | conflict |
PDB | External Database | Details |
---|---|---|
Arg 376 | - | expression tag |
Phe 377 | - | expression tag |
Arg 378 | - | expression tag |
Leu 379 | - | expression tag |
Gly 380 | - | expression tag |
Phe 381 | - | expression tag |
Met 382 | - | expression tag |
Ala 383 | - | expression tag |
Thr 384 | - | expression tag |
Phe 385 | - | expression tag |
Pro 386 | - | expression tag |
Cys 387 | - | expression tag |
Cys 388 | - | expression tag |
Pro 389 | - | expression tag |
Asn 390 | - | expression tag |
Pro 391 | - | expression tag |
Gly 392 | - | expression tag |
Pro 393 | - | expression tag |
Pro 394 | - | expression tag |
Gly 395 | - | expression tag |
Ala 396 | - | expression tag |
Arg 397 | - | expression tag |
Gly 398 | - | expression tag |
Glu 399 | - | expression tag |
Val 400 | - | expression tag |
Gly 401 | - | expression tag |
Glu 402 | - | expression tag |
Glu 403 | - | expression tag |
Glu 404 | - | expression tag |
Glu 405 | - | expression tag |
Gly 406 | - | expression tag |
Glu 407 | - | expression tag |
Phe 408 | - | expression tag |
Leu 409 | - | expression tag |
Glu 410 | - | expression tag |
Val 411 | - | expression tag |
Leu 412 | - | expression tag |
Phe 413 | - | expression tag |
Gln 414 | - | expression tag |
Gly 415 | - | expression tag |
Pro 416 | - | expression tag |
His 417 | - | expression tag |
His 418 | - | expression tag |
His 419 | - | expression tag |
His 420 | - | expression tag |
His 421 | - | expression tag |
His 422 | - | expression tag |
His 423 | - | expression tag |
His 424 | - | expression tag |
His 425 | - | expression tag |
His 426 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 60450.4 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 411.9 | |
All* | Total formula weight | 60862.2 |