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7BCM

The DDR1 Kinase Domain Bound To SR302

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, BEpithelial discoidin domain-containing receptor 1polymer31535754.12UniProt (Q08345)
Pfam (PF07714)
In PDB
Homo sapiens (Human)Epithelial discoidin domain receptor 1,CD167 antigen-like family member A,Cell adhesion kinase,Discoidin receptor tyrosine kinase,HGK2,Mammary carcinoma kinase 10,MCK-10,Protein-tyrosine kinase 3A,Protein-tyrosine kinase RTK-6,TRK E,Tyrosine kinase DDR,Tyrosine-protein kinase CAK
2A, B~{N}-[[4-[[(2~{S})-4-cyclohexyl-1-[[(3~{S})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamidenon-polymer622.82Chemie (TBK)
3waterwater18.021Chemie (HOH)
Sequence modifications
A, B: 601 - 913 (UniProt: Q08345)
PDBExternal DatabaseDetails
Ser 599-expression tag
Met 600-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight71508.2
Non-Polymers*Number of molecules2
Total formula weight1245.6
All*Total formula weight72753.7
*Water molecules are not included.

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PDB entries from 2024-07-10

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