6F1W
Crystal structure of human Casein Kinase I delta in complex with compound 31a
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Casein kinase I isoform delta | polymer | 314 | 36457.9 | 1 | UniProt (P48730) Pfam (PF00069) In PDB | Homo sapiens (Human) | CKId,Tau-protein kinase CSNK1D |
2 | B | Casein kinase I isoform delta | polymer | 314 | 36377.9 | 1 | UniProt (P48730) Pfam (PF00069) In PDB | Homo sapiens (Human) | CKId,Tau-protein kinase CSNK1D |
3 | A, B | SULFATE ION | non-polymer | 96.1 | 15 | Chemie (SO4) | |||
4 | A, B | (9~{R},10~{R},11~{S})-~{N}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | non-polymer | 623.7 | 2 | Chemie (CG5) | |||
5 | water | water | 18.0 | 415 | Chemie (HOH) |
Sequence modifications
A: 1 - 294 (UniProt: P48730)
B: 1 - 294 (UniProt: P48730)
PDB | External Database | Details |
---|---|---|
Met -19 | - | initiating methionine |
Gly -18 | - | expression tag |
Ser -17 | - | expression tag |
Ser -16 | - | expression tag |
His -15 | - | expression tag |
His -14 | - | expression tag |
His -13 | - | expression tag |
His -12 | - | expression tag |
His -11 | - | expression tag |
His -10 | - | expression tag |
Ser -9 | - | expression tag |
Ser -8 | - | expression tag |
Gly -7 | - | expression tag |
Leu -6 | - | expression tag |
Val -5 | - | expression tag |
Pro -4 | - | expression tag |
Arg -3 | - | expression tag |
Gly -2 | - | expression tag |
Ser -1 | - | expression tag |
His 0 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Met -19 | - | initiating methionine |
Gly -18 | - | expression tag |
Ser -17 | - | expression tag |
Ser -16 | - | expression tag |
His -15 | - | expression tag |
His -14 | - | expression tag |
His -13 | - | expression tag |
His -12 | - | expression tag |
His -11 | - | expression tag |
His -10 | - | expression tag |
Ser -9 | - | expression tag |
Ser -8 | - | expression tag |
Gly -7 | - | expression tag |
Leu -6 | - | expression tag |
Val -5 | - | expression tag |
Pro -4 | - | expression tag |
Arg -3 | - | expression tag |
Gly -2 | - | expression tag |
Ser -1 | - | expression tag |
His 0 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 72835.8 | |
Non-Polymers* | Number of molecules | 17 |
Total formula weight | 2688.3 | |
All* | Total formula weight | 75524.0 |