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6DQ7

LINKED KDM5A JMJ DOMAIN BOUND TO THE POTENTIAL HYDROLYSIS PRODUCT OF INHIBITOR N45 i.e. 3-((6-(4-(2-cyano-3-methylbut-2-enoyl)-1,4-diazepan-1-yl)-2-(pyridin-2-yl)pyrimidin-4-yl)amino)propanoic acid

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1ALinked KDM5A Jmj Domainpolymer33037944.81UniProt (P29375)
Pfam (PF02375)
Pfam (PF02373)
In PDB
Homo sapiens (Human)Histone demethylase JARID1A,Jumonji/ARID domain-containing protein 1A,Retinoblastoma-binding protein 2,RBBP-2,Histone demethylase JARID1A,Jumonji/ARID domain-containing protein 1A,Retinoblastoma-binding protein 2,RBBP-2
2AN-{6-[4-(hydroxyacetyl)-1,4-diazepan-1-yl]-2-(pyridin-2-yl)pyrimidin-4-yl}-beta-alaninenon-polymer400.41Chemie (H6M)
3AMANGANESE (II) IONnon-polymer54.91Chemie (MN)
4A1,2-ETHANEDIOLnon-polymer62.11Chemie (EDO)
5AGLYCEROLnon-polymer92.11Chemie (GOL)
6waterwater18.0202Chemie (HOH)
Sequence modifications
A: 1 - 347 (UniProt: P29375)
PDBExternal DatabaseDetails
His -1-expression tag
Asn 0-expression tag
A: 348 - 588 (UniProt: P29375)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight37944.8
Non-Polymers*Number of molecules4
Total formula weight609.5
All*Total formula weight38554.4
*Water molecules are not included.

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PDB entries from 2024-03-27

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