5NGB
X-Ray Diffraction Crystal Structure of the murine PI3K p110delta in complex with a pan inhibitor
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | polymer | 1079 | 124313.1 | 1 | UniProt (Q3UDT3) Pfam (PF02192) Pfam (PF00794) Pfam (PF00792) Pfam (PF00613) Pfam (PF00454) UniProt (by SIFTS) (O35904) In PDB | Mus musculus (House Mouse) | Putative uncharacterized protein |
2 | A | 3-[[4-(2-morpholin-4-yl-4-oxidanylidene-3~{H}-quinolin-8-yl)-1,2,3-triazol-1-yl]methyl]benzoic acid | non-polymer | 431.4 | 1 | Chemie (8WH) |
Sequence modifications
A: -6 - 1044 (UniProt: Q3UDT3)
PDB | External Database | Details |
---|---|---|
Met -34 | - | initiating methionine |
Ser -33 | - | expression tag |
Tyr -32 | - | expression tag |
Tyr -31 | - | expression tag |
His -30 | - | expression tag |
His -29 | - | expression tag |
His -28 | - | expression tag |
His -27 | - | expression tag |
His -26 | - | expression tag |
His -25 | - | expression tag |
Asp -24 | - | expression tag |
Tyr -23 | - | expression tag |
Asp -22 | - | expression tag |
Ile -21 | - | expression tag |
Pro -20 | - | expression tag |
Thr -19 | - | expression tag |
Thr -18 | - | expression tag |
Glu -17 | - | expression tag |
Asn -16 | - | expression tag |
Leu -15 | - | expression tag |
Tyr -14 | - | expression tag |
Phe -13 | - | expression tag |
Gln -12 | - | expression tag |
Gly -11 | - | expression tag |
Ala -10 | - | expression tag |
Met -9 | - | expression tag |
Asp -8 | - | expression tag |
Leu -7 | - | expression tag |
Glu 99 | - | insertion |
Asn 100 | - | insertion |
Leu 101 | - | insertion |
Tyr 102 | - | insertion |
Phe 103 | - | insertion |
Gln 104 | - | insertion |
Gly 105 | - | insertion |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 124313.1 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 431.4 | |
All* | Total formula weight | 124744.5 |