5M25
Modulation of MLL1 Methyltransferase Activity
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A | WD repeat-containing protein 5 | polymer | 434 | 48112.3 | 1 | UniProt (P61964) Pfam (PF00400) In PDB | Homo sapiens (Human) | BMP2-induced 3-kb gene protein |
2 | A | (2~{S})-2-[[(2~{S})-2-[[(2~{S})-2-azanyl-3-oxidanyl-propanoyl]amino]propanoyl]amino]-5-carbamimidamido-~{N}-[(2~{S})-1-[[4-[(~{E})-[4-(hydroxymethyl)phenyl]diazenyl]phenyl]methylamino]-1-oxidanylidene-propan-2-yl]pentanamide | non-polymer | 626.7 | 1 | Chemie (7DU) | |||
3 | water | water | 18.0 | 98 | Chemie (HOH) |
Sequence modifications
A: 22 - 334 (UniProt: P61964)
PDB | External Database | Details |
---|---|---|
Met -99 | - | initiating methionine |
Gly -98 | - | expression tag |
Ser -97 | - | expression tag |
Ser -96 | - | expression tag |
His -95 | - | expression tag |
His -94 | - | expression tag |
His -93 | - | expression tag |
His -92 | - | expression tag |
His -91 | - | expression tag |
His -90 | - | expression tag |
Ser -89 | - | expression tag |
Ser -88 | - | expression tag |
Gly -87 | - | expression tag |
Leu -86 | - | expression tag |
Val -85 | - | expression tag |
Pro -84 | - | expression tag |
Arg -83 | - | expression tag |
Gly -82 | - | expression tag |
Ser -81 | - | expression tag |
His -80 | - | expression tag |
Met -79 | - | expression tag |
Ala -78 | - | expression tag |
Ser -77 | - | expression tag |
Met -76 | - | expression tag |
Ser -75 | - | expression tag |
Asp -74 | - | expression tag |
Ser -73 | - | expression tag |
Glu -72 | - | expression tag |
Val -71 | - | expression tag |
Asn -70 | - | expression tag |
Gln -69 | - | expression tag |
Glu -68 | - | expression tag |
Ala -67 | - | expression tag |
Lys -66 | - | expression tag |
Pro -65 | - | expression tag |
Glu -64 | - | expression tag |
Val -63 | - | expression tag |
Lys -62 | - | expression tag |
Pro -61 | - | expression tag |
Glu -60 | - | expression tag |
Val -59 | - | expression tag |
Lys -58 | - | expression tag |
Pro -57 | - | expression tag |
Glu -56 | - | expression tag |
Thr -55 | - | expression tag |
His -54 | - | expression tag |
Ile -53 | - | expression tag |
Asn -52 | - | expression tag |
Leu -51 | - | expression tag |
Lys -50 | - | expression tag |
Val -49 | - | expression tag |
Ser -48 | - | expression tag |
Asp -47 | - | expression tag |
Gly -46 | - | expression tag |
Ser -45 | - | expression tag |
Ser -44 | - | expression tag |
Glu -43 | - | expression tag |
Ile -42 | - | expression tag |
Phe -41 | - | expression tag |
Phe -40 | - | expression tag |
Lys -39 | - | expression tag |
Ile -38 | - | expression tag |
Lys -37 | - | expression tag |
Lys -36 | - | expression tag |
Thr -35 | - | expression tag |
Thr -34 | - | expression tag |
Pro -33 | - | expression tag |
Leu -32 | - | expression tag |
Arg -31 | - | expression tag |
Arg -30 | - | expression tag |
Leu -29 | - | expression tag |
Met -28 | - | expression tag |
Glu -27 | - | expression tag |
Ala -26 | - | expression tag |
Phe -25 | - | expression tag |
Ala -24 | - | expression tag |
Lys -23 | - | expression tag |
Arg -22 | - | expression tag |
Gln -21 | - | expression tag |
Gly -20 | - | expression tag |
Lys -19 | - | expression tag |
Glu -18 | - | expression tag |
Met -17 | - | expression tag |
Asp -16 | - | expression tag |
Ser -15 | - | expression tag |
Leu -14 | - | expression tag |
Arg -13 | - | expression tag |
Phe -12 | - | expression tag |
Leu -11 | - | expression tag |
Tyr -10 | - | expression tag |
Asp -9 | - | expression tag |
Gly -8 | - | expression tag |
Ile -7 | - | expression tag |
Arg -6 | - | expression tag |
Ile -5 | - | expression tag |
Gln -4 | - | expression tag |
Ala -3 | - | expression tag |
Asp -2 | - | expression tag |
Gln -1 | - | expression tag |
Thr 0 | - | expression tag |
Pro 1 | - | expression tag |
Glu 2 | - | expression tag |
Asp 3 | - | expression tag |
Leu 4 | - | expression tag |
Asp 5 | - | expression tag |
Met 6 | - | expression tag |
Glu 7 | - | expression tag |
Asp 8 | - | expression tag |
Asn 9 | - | expression tag |
Asp 10 | - | expression tag |
Ile 11 | - | expression tag |
Ile 12 | - | expression tag |
Glu 13 | - | expression tag |
Ala 14 | - | expression tag |
His 15 | - | expression tag |
Arg 16 | - | expression tag |
Glu 17 | - | expression tag |
Gln 18 | - | expression tag |
Ile 19 | - | expression tag |
Gly 20 | - | expression tag |
Gly 21 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 48112.3 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 626.7 | |
All* | Total formula weight | 48739.0 |