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5G4R

BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-dimethyl-6-2R-2- methylpiperazin-1-yl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl-2- methoxybenzamide

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B, C, DPEREGRINpolymer11813925.94UniProt (P55201)
Pfam (PF00439)
In PDB
HOMO SAPIENS (HUMAN)BROMODOMAIN AND PHD FINGER-CONTAINING PROTEIN 1, PROTEIN BR140,
2A, B, C, DN-[1,3-dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxidanylidene-benzimidazol-5-yl]-2-methoxy-benzamidenon-polymer409.54Chemie (LF1)
3waterwater18.0400Chemie (HOH)
Sequence modifications
A, B, C, D: 622 - 738 (UniProt: P55201)
PDBExternal DatabaseDetails
Gly 621-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight55703.7
Non-Polymers*Number of molecules4
Total formula weight1637.9
All*Total formula weight57341.6
*Water molecules are not included.

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PDB entries from 2024-05-15

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