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5DXH

p110alpha/p85alpha with compound 5

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, DPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformpolymer1067124313.82UniProt (P42336)
Pfam (PF02192)
Pfam (PF00794)
Pfam (PF00792)
Pfam (PF00613)
Pfam (PF00454)
In PDB
Homo sapiens (Human)PtdIns-3-kinase subunit alpha,Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha,p110alpha,Phosphoinositide-3-kinase catalytic alpha polypeptide,Serine/threonine protein kinase PIK3CA
2B, EPhosphatidylinositol 3-kinase regulatory subunit alphapolymer16920879.62UniProt (P23727)
Pfam (PF16454)
In PDB
Bos taurus (Bovine)PtdIns-3-kinase regulatory subunit alpha,Phosphatidylinositol 3-kinase 85 kDa regulatory subunit alpha,PtdIns-3-kinase regulatory subunit p85-alpha
3A, Dmethyl {2-[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamatenon-polymer452.92Chemie (5H2)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight290386.7
Non-Polymers*Number of molecules2
Total formula weight905.8
All*Total formula weight291292.5
*Water molecules are not included.

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PDB entries from 2024-05-08

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